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Pharmaceutical Sciences Experts

Mai Antonello


Chemistry and Technology of Drugs
La Sapienza University
Italy

Biography

MAI Antonello is working in the department of Chemistry and Technology of Drugs at La Sapienza University, Italy. 

Research Interest

Pharmaceutical area

Publications

  • Binda C, Valente S, Romanenghi M, Pilotto S, Cirilli R, Karytinos A, Ciossani G, Botrugno OA, Forneris F, Tardugno M, Edmondson DE. Biochemical, structural, and biological evaluation of tranylcypromine derivatives as inhibitors of histone demethylases LSD1 and LSD2. Journal of the American Chemical Society. 2010 Apr 23;132(19):6827-33.

  • Mai A, Valente S, Cheng D, Perrone A, Ragno R, Simeoni S, Sbardella G, Brosch G, Nebbioso A, Conte M, Altucci L. Synthesis and biological validation of novel synthetic histone/protein methyltransferase inhibitors. ChemMedChem. 2007 Jul 9;2(7):987-91.

  • Mai A, Massa S, Rotili D, Cerbara I, Valente S, Pezzi R, Simeoni S, Ragno R. Histone deacetylation in epigenetics: an attractive target for anticancer therapy. Medicinal research reviews. 2005 May 1;25(3):261-309.

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